Gamba, IlariaSalvadó, IriaBrissos, Rosa F.Gamez, PatrickBrea Floriani, José ManuelLoza García, María IsabelVázquez Sentís, Marco EugenioVázquez López, Miguel2018-07-132018-07-132016Gamba, I., Salvadó, I., Brissos, R., Gamez, P., Brea, J., & Loza, M. et al. (2016). High-affinity sequence-selective DNA binding by iridium(iii) polypyridyl organometallopeptides. Chemical Communications, 52(6), 1234-1237. doi: 10.1039/c5cc07619f1359-7345http://hdl.handle.net/10347/17021We demonstrate the application of solid-phase peptide synthesis methods for the straightforward assembly of polynuclear Ir(III) organometallopeptides, and show that their oligoarginine derivatives exhibit high DNA binding affinity, sequence selectivity, and high cytotoxicity towards a set of cancer cell lineseng© The Royal Society of Chemistry 2016High-affinity sequence-selective DNA binding by iridium(III) polypyridyl organometallopeptidesjournal article10.1039/C5CC07619F1364-548Xopen access